產品屬性:
產品名稱 | Obafistat |
規格 | 10mM*1 mL in DMSO、5 mg、10 mg、50 mg |
貨號 | EY-01Y18086 |
Cas No.: 2160582-57-8
別名: N/A
化學名: N/A
分子式: C15H16FN5O3S
分子量: 365.38
溶解度: DMSO : 62.5 mg/mL (171.05 mM; ultrasonic and warming and heat to 60°C)
儲存條件: 4°C, protect from light
General tips:For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition:Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述:
Obafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4)[1].[1]. Marcus Koppitz, et al. [8-(phenylsulfonyl)-3,8-diazabicyclo[3.2.1]oct-3-yl] (1h-1,2,3-triazol-4-yl)methanones. WO2017202817A1.
特別提醒公司產品僅供科研使用